SCHEMBL9514348

SCHEMBL9514348

CC(C)c1cc(-c2ccccc2)cc(-c2ccc(F)cc2)c1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
PTPN1 P18031 1/20 0.44
HMGCR P04035 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
BACE1 P56817 1/20 0.39
PTPN5 P54829 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
BCL2 P10415 1/20 0.37
MCL1 Q07820 1/20 0.37
ALOX5 P09917 1/20 0.37
HSP90AA1 P07900 1/20 0.37
AKR1C2 P52895 2/20 0.36
AKR1C1 Q04828 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9512239 0.94 CA1 (0.53) CA1CA2HMGCRGABRA1GABRB1
SCHEMBL31603747 0.91 CA1 (0.57) CA1CA2PTPN1GABRA1GABRB1
SCHEMBL10026552 0.84 CA1 (0.68) CA1CA2HMGCRGABRA1GABRB1
SCHEMBL9857638 0.82 HMGCR (0.42) HMGCRGABRA1
SCHEMBL9196802 0.82 HMGCR (0.39) HMGCRAKR1C2AKR1C1PTGS1PTGS2
SCHEMBL10026544 0.82 CA1 (0.71) CA1CA2GABRA1GABRB1ALDH1A1
SCHEMBL9857543 0.81 HMGCR (0.44) PTPN1HMGCRAKR1C2AKR1C1PTGS1
SCHEMBL9194475 0.80 HMGCR (0.45) CA1CA2PTPN1HMGCRGABRA1
SCHEMBL24757582 0.80 CA1 (0.74) CA1CA2GABRA1GABRB1ALDH1A1
SCHEMBL8780176 0.80 GABRA1 (0.50) CA1CA2HMGCRGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0341681-B1 6-Phenoxymethyl-4-hydroxytetrahydropyran-2-ones and 6-thiophenoxymethyl-4-hydroxytetrahydropyran-2-ones, the corresponding dihydrocarboxylic-acid derivatives, salts and esters, process for preparing these compounds, their use as medicines, pharmaceutical compositions and phenols and thiophenols HOECHST AG (DE) 1993-12-29 EP disclosed
US-5166171-A Compounds for treatment of artheriosclerosis and hypercholesterolemia HOECHST AKTIENGESELLSCHAFT (DE) 1992-11-24 US disclosed
EP-0341681-A2 6-Phenoxymethyl-4-hydroxytetrahydropyran-2-ones and 6-thiophenoxymethyl-4-hydroxytetrahydropyran-2-ones, the corresponding dihydrocarboxylic-acid derivatives, salts and esters, process for preparing these compounds, their use as medicines, pharmaceutical compositions and phenols and thiophenols HOECHST AKTIENGESELLSCHAFT (DE) 1989-11-15 EP disclosed