SCHEMBL9512239

SCHEMBL9512239

CC(C)c1cc(-c2ccc(F)cc2)cc(-c2ccc(F)cc2)c1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
HMGCR P04035 2/20 0.44
GCGR P47871 2/20 0.39
RPS6KA3 P51812 3/20 0.39
GSK3B P49841 1/20 0.38
GABRA1 P14867 5/20 0.37
GABRB1 P18505 4/20 0.37
GABRB2 P47870 3/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
IKBKB O14920 1/20 0.35
CHUK O15111 1/20 0.35
FAAH O00519 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
GABRG2 P18507 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9514348 0.94 CA1 (0.47) CA1CA2HMGCRGABRA1GABRB1
SCHEMBL10026552 0.89 CA1 (0.68) CA1CA2HMGCRGCGRRPS6KA3
SCHEMBL8780176 0.85 GABRA1 (0.50) CA1CA2HMGCRGCGRRPS6KA3
SCHEMBL22888675 0.84 CA1 (0.55) CA1CA2HMGCRGCGRRPS6KA3
SCHEMBL9199239 0.83 CA1 (0.41) CA1CA2HMGCRGCGRRPS6KA3
SCHEMBL31603747 0.82 CA1 (0.57) CA1CA2GABRA1GABRB1GABRB2
SCHEMBL9516053 0.81 CA1 (0.39) CA1CA2
SCHEMBL9197287 0.80 HMGCR (0.38) CA1CA2HMGCRGCGRRPS6KA3
SCHEMBL8780227 0.80 HMGCR (0.50) CA1CA2HMGCRGCGRRPS6KA3
SCHEMBL9514015 0.79 HMGCR (0.42) CA1CA2HMGCRGCGRIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0341681-B1 6-Phenoxymethyl-4-hydroxytetrahydropyran-2-ones and 6-thiophenoxymethyl-4-hydroxytetrahydropyran-2-ones, the corresponding dihydrocarboxylic-acid derivatives, salts and esters, process for preparing these compounds, their use as medicines, pharmaceutical compositions and phenols and thiophenols HOECHST AG (DE) 1993-12-29 EP disclosed
US-5166171-A Compounds for treatment of artheriosclerosis and hypercholesterolemia HOECHST AKTIENGESELLSCHAFT (DE) 1992-11-24 US disclosed
EP-0341681-A2 6-Phenoxymethyl-4-hydroxytetrahydropyran-2-ones and 6-thiophenoxymethyl-4-hydroxytetrahydropyran-2-ones, the corresponding dihydrocarboxylic-acid derivatives, salts and esters, process for preparing these compounds, their use as medicines, pharmaceutical compositions and phenols and thiophenols HOECHST AKTIENGESELLSCHAFT (DE) 1989-11-15 EP disclosed