SCHEMBL9197367

SCHEMBL9197367

CC(=O)Nc1ncc(C(C)=O)cc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
POLB P06746 1/20 0.40
NPC1 O15118 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 2/20 0.40
KCNH2 Q12809 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
RAB9A P51151 2/20 0.39
DYRK1A Q13627 1/20 0.38
TP53 P04637 1/20 0.37
ADORA3 P0DMS8 2/20 0.36
HTT P42858 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTK2 Q05397 1/20 0.34
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25684289 0.84 SMN1; SMN2 (0.36) ALDH1A1POLBNPC1SMN1; SMN2MAPT
SCHEMBL11637557 0.82 MAPT (0.51) ALDH1A1POLBNPC1SMN1; SMN2MAPT
SCHEMBL7091347 0.81 MAPT (0.47) ALDH1A1POLBNPC1SMN1; SMN2MAPT
SCHEMBL7091354 0.81 L3MBTL1 (0.40) ALDH1A1POLBNPC1SMN1; SMN2L3MBTL1
SCHEMBL9198708 0.79 ALDH1A1 (0.44) ALDH1A1POLBNPC1SMN1; SMN2MAPT
SCHEMBL9995068 0.79 PTK2 (0.49) ALDH1A1POLBNPC1SMN1; SMN2MAPT
SCHEMBL21597026 0.79 L3MBTL1 (0.39) POLBNPC1SMN1; SMN2MAPTKCNH2
SCHEMBL913171 0.79 L3MBTL1 (0.39) ALDH1A1NPC1SMN1; SMN2MAPTKCNH2
SCHEMBL9193957 0.76 CA5A (0.37) ALDH1A1POLBNPC1SMN1; SMN2RAB9A
SCHEMBL914646 0.74 GAA (0.54) ALDH1A1SMN1; SMN2MAPTPKMDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299277-B1 Process for the preparation of substituted pyridyl-alkyl ketones BAYER AG (DE) 1995-10-18 EP disclosed
US-4990620-A Halogen substituted pyridylalkyl ketones BAYER AKTIENGESELLSCHAFT (DE) 1991-02-05 US disclosed
US-4927938-A Halogen substituted pyridylalkyl ketones BAYER AKTIENGESELLSCHAFT (DE) 1990-05-22 US disclosed
EP-0299277-A2 Process for the preparation of substituted pyridyl-alkyl ketones BAYER AG (DE) 1989-01-18 EP disclosed