SCHEMBL9197865

SCHEMBL9197865

CCCCC(OC(=O)c1c[nH]c2ncccc12)C1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.51
CNR2 P34972 1/20 0.39
BCHE P06276 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CCNE1 P24864 4/20 0.37
CDK2 P24941 4/20 0.37
HSD11B1 P28845 3/20 0.36
ADORA2A P29274 1/20 0.36
PIM1 P11309 1/20 0.36
PIM3 Q86V86 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
CDC7 O00311 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKACA P17612 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CDK8 P49336 1/20 0.35
CLK2 P49760 1/20 0.35
CDK5 Q00535 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3166028 0.73 HTR4 (0.51) CYP2D6
SCHEMBL9539487 0.73 HTR3E (0.44) CYP2D6
Hydrochloric Acid SCHEMBL9340476 0.72 APEX1 (0.45) CYP2D6
SCHEMBL858042 0.71 HTR3E (0.63) MAP2K1CNR2CYP2D6CYP2C9CYP2C19
SCHEMBL7956049 0.70 MAP2K1 (0.74) MAP2K1CNR2ADORA2AMTNR1A
SCHEMBL29526844 0.70 MAP2K1 (1.00) MAP2K1CNR2ADORA2AMTNR1AAXL
SCHEMBL1607007 0.70 MAP2K1 (1.00) MAP2K1CNR2ADORA2AMTNR1AAXL
SCHEMBL7393472 0.69 HTR4 (0.58) MAP2K1
SCHEMBL9280928 0.69 ALDH1A1 (0.31)
SCHEMBL3165607 0.68 HTR3E (0.41) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662959-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-07-19 EP disclosed