SCHEMBL9198136

SCHEMBL9198136

COc1ccc(C2(O)CCC(CCN3CCN(c4ccccn4)CC3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.59
DRD2 P14416 3/20 0.53
DRD3 P35462 2/20 0.53
SIGMAR1 Q99720 1/20 0.52
LMNA P02545 2/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.48
HPGD P15428 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9198134 1.00 HTR1A (0.59) HTR1ADRD2DRD3SIGMAR1LMNA
SCHEMBL9197517 1.00 HTR1A (0.59) HTR1ADRD2DRD3SIGMAR1LMNA
SCHEMBL9195870 0.89 DRD2 (0.59) HTR1ADRD2DRD3POLB
SCHEMBL9200413 0.87 DRD2 (0.55) HTR1ADRD2DRD3SIGMAR1LMNA
SCHEMBL9202549 0.83 DRD2 (0.55) HTR1ADRD2DRD3
SCHEMBL9202889 0.83 HTR1A (0.57) HTR1ALMNAALDH1A1KMT2AHPGD
SCHEMBL9196526 0.82 DRD2 (0.59) HTR1ADRD2DRD3SIGMAR1
SCHEMBL9196967 0.81 DRD2 (0.53) HTR1ADRD2DRD3SIGMAR1
SCHEMBL9197205 0.78 DRD2 (0.62) HTR1ADRD2DRD3SIGMAR1
SCHEMBL9197201 0.78 DRD2 (0.62) HTR1ADRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed