SCHEMBL9200413

SCHEMBL9200413

OC1(c2ccc(F)cc2)CCC(CCN2CCN(c3ccccn3)CC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.55
DRD3 P35462 10/20 0.55
HTR1A P08908 6/20 0.55
HTR2A P28223 6/20 0.55
HTR7 P34969 6/20 0.55
DRD4 P21917 6/20 0.55
SIGMAR1 Q99720 4/20 0.55
SLC6A4 P31645 3/20 0.55
HTR2C P28335 2/20 0.55
GRIN2B Q13224 1/20 0.54
ADRA2C P18825 3/20 0.53
DRD1 P21728 3/20 0.53
DRD5 P21918 3/20 0.53
HRH1 P35367 3/20 0.53
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9195870 0.91 DRD2 (0.59) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL9197517 0.87 HTR1A (0.59) DRD2DRD3HTR1ASIGMAR1LMNA
SCHEMBL9198136 0.87 HTR1A (0.59) DRD2DRD3HTR1ASIGMAR1LMNA
SCHEMBL9198134 0.87 HTR1A (0.59) DRD2DRD3HTR1ASIGMAR1LMNA
SCHEMBL9202549 0.85 DRD2 (0.55) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL9196526 0.85 DRD2 (0.59) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL9196967 0.84 DRD2 (0.53) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL29974343 0.81 GRIN2B (0.66) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL22626906 0.81 GRIN2B (0.66) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL9197205 0.80 DRD2 (0.62) DRD2DRD3HTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4975445-A Antidepressants WARNER-LAMBERT COMPANY (US) 1990-12-04 US disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed