SCHEMBL9199035

SCHEMBL9199035

CCc1cc(-c2cccc(CC)c2O)ccc1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.60
PTPN5 P54829 1/20 0.54
GABRA1 P14867 1/20 0.53
GABRB2 P47870 1/20 0.53
HSD17B1 P14061 3/20 0.50
ESR1 P03372 4/20 0.47
ESR2 Q92731 4/20 0.47
HSD17B2 P37059 1/20 0.46
ALOX5 P09917 1/20 0.44
AR P10275 1/20 0.42
ANPEP P15144 1/20 0.42
DPP4 P27487 1/20 0.42
APP P05067 1/20 0.41
BACE1 P56817 1/20 0.41
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
PDK2 Q15119 1/20 0.39
MCL1 Q07820 1/20 0.38
DAO P14920 1/20 0.37
DDO Q99489 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3558975 0.86 HSD17B1 (0.53) AKR1B1PTPN5GABRA1GABRB2HSD17B1
SCHEMBL9198775 0.83 ALOX5 (0.60) AKR1B1PTPN5GABRA1GABRB2ESR1
SCHEMBL10454627 0.80 GABRA1 (0.59) AKR1B1PTPN5GABRA1GABRB2HSD17B1
SCHEMBL16581416 0.80 HSD17B1 (0.62) GABRA1GABRB2HSD17B1ESR1ESR2
SCHEMBL3953461 0.79 HSD17B1 (0.71) GABRA1GABRB2HSD17B1ESR1ESR2
SCHEMBL16527783 0.79 GABRA1 (0.76) PTPN5GABRA1GABRB2ANPEPDPP4
SCHEMBL10911038 0.78 GABRA1 (0.61) PTPN5GABRA1GABRB2ANPEPDPP4
SCHEMBL13678958 0.77 HSD17B1 (0.75) GABRA1GABRB2HSD17B1ESR1ESR2
SCHEMBL4907630 0.76 AKR1B1 (1.00) AKR1B1GABRA1GABRB2ALOX5
SCHEMBL2030094 0.76 TLR8 (0.49) AKR1B1PTPN5GABRA1GABRB2HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0382213-B1 Biphenyl derivative, nerve cell degeneration repairing or protecting agent and process for preparing a phenyl derivative contained in the agent OTSUKA PHARMA CO LTD (JP) 1995-05-10 EP disclosed
US-5053548-A Containing hydroxy substituents; nervous system disorders OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1991-10-01 US disclosed
EP-0382213-A2 Biphenyl derivative, nerve cell degeneration repairing or protecting agent and process for preparing a phenyl derivative contained in the agent OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed