SCHEMBL9199064

SCHEMBL9199064

CC(=O)Oc1nn(Cc2ccc(Br)cc2F)c(=O)c2ncccc12

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 6/20 0.67
MEN1 O00255 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
KMT2A Q03164 1/20 0.52
HSD17B10 Q99714 1/20 0.52
BRD4 O60885 2/20 0.42
KDM4E B2RXH2 1/20 0.39
P2RX7 Q99572 2/20 0.38
MAPT P10636 1/20 0.37
PTGER1 P34995 1/20 0.37
RORC P51449 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9205172 0.92 AKR1B1 (0.62) AKR1B1MEN1CYP1A2CYP2C9KMT2A
SCHEMBL9870990 0.88 AKR1B1 (0.62) AKR1B1MEN1CYP1A2CYP2C9KMT2A
SCHEMBL9872250 0.81 AKR1B1 (0.57) AKR1B1MEN1CYP1A2CYP2C9KMT2A
SCHEMBL9209897 0.77 AKR1B1 (0.85) AKR1B1MEN1CYP1A2CYP2C9KMT2A
SCHEMBL9206818 0.72 AKR1B1 (0.57) AKR1B1MEN1KMT2ABRD4
SCHEMBL9201378 0.71 AKR1B1 (0.57) AKR1B1MEN1CYP1A2CYP2C9KMT2A
SCHEMBL9204791 0.70 AKR1B1 (0.71) AKR1B1
SCHEMBL11165597 0.69 AKR1B1 (0.77) AKR1B1MEN1CYP1A2CYP2C9KMT2A
SCHEMBL9207611 0.69 AKR1B1 (0.54) AKR1B1MEN1CYP1A2CYP2C9KMT2A
Ponalrestat SCHEMBL49154 0.68 AKR1B1 (1.00) AKR1B1MEN1CYP1A2CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0401981-B1 Pyridazinone deriratives PFIZER (US) 1995-04-26 EP disclosed