SCHEMBL9199191

SCHEMBL9199191

CCOC(=O)CCCc1ccc2c(c1)CC(N)CC2

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.47
DRD2 P14416 3/20 0.44
DRD3 P35462 3/20 0.44
BRD4 O60885 1/20 0.43
CYP4Z1 Q86W10 2/20 0.42
CYP4F11 Q9HBI6 1/20 0.42
CYP4F12 Q9HCS2 1/20 0.42
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP4F2 P78329 2/20 0.41
CYP4A11 Q02928 2/20 0.41
ALOX5 P09917 1/20 0.40
SMYD3 Q9H7B4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9134280 0.99 ACHE (0.47) ACHEDRD2DRD3BRD4CYP4Z1
SCHEMBL9195127 0.93 ACHE (0.49) ACHEDRD2DRD3CYP4F2CYP4A11
SCHEMBL5679141 0.93 ACHE (0.49) ACHEDRD2DRD3CYP4F2CYP4A11
SCHEMBL9191715 0.93 ACHE (0.49) ACHEDRD2DRD3CYP4F2CYP4A11
Hydrochloric Acid SCHEMBL9133231 0.92 ACHE (0.48) ACHEDRD2DRD3CYP4Z1CYP4F2
Hydrochloric Acid SCHEMBL9133151 0.92 ACHE (0.48) ACHEDRD2DRD3CYP4Z1CYP4F2
Hydrochloric Acid SCHEMBL9133223 0.92 ACHE (0.48) ACHEDRD2DRD3CYP4Z1CYP4F2
SCHEMBL9305655 0.84 BRD4 (0.60) ACHEDRD2DRD3BRD4
SCHEMBL9305716 0.83 BRD4 (0.56) ACHEDRD2DRD3BRD4
Hydrochloric Acid SCHEMBL9304134 0.83 BRD4 (0.58) ACHEDRD2DRD3BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0500443-B1 Phenylethanolamino- and phenylethanolaminomethyltetralines, process for their preparation, intermediates of this process and pharmaceutical compositions containing them SANOFI SA (FR) 1995-04-26 EP disclosed
EP-0500443-A1 Phenylethanolamino- and phenylethanolaminomethyltetralines, process for their preparation, intermediates of this process and pharmaceutical compositions containing them SANOFI (FR) 1992-08-26 EP disclosed
EP-0499755-A1 Phenylethanolaminotetralines, process for their preparation, intermediates of this process and pharmaceutical compositions containing them MIDY S.p.A. (IT) 1992-08-26 EP disclosed