SCHEMBL9199725

SCHEMBL9199725

O=C(NC1CCC(CN2CCN(c3ccccn3)CC2)CC1)c1ccccc1

nearest known ligand 0.81

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.81
DRD3 P35462 5/20 0.60
ALDH1A1 P00352 3/20 0.58
HTR1A P08908 3/20 0.54
HTR2A P28223 3/20 0.53
POLB P06746 1/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199135 0.89 DRD2 (1.00) DRD2DRD3ALDH1A1HTR1AHTR2A
SCHEMBL9195887 0.88 DRD2 (0.64) DRD2DRD3ALDH1A1
SCHEMBL8172030 0.83 DRD2 (0.80) DRD2DRD3ALDH1A1POLB
SCHEMBL8172032 0.83 DRD2 (0.80) DRD2DRD3ALDH1A1POLB
SCHEMBL13648727 0.82 DRD2 (0.62) DRD2DRD3ALDH1A1HTR1AHTR2A
SCHEMBL9200670 0.82 DRD2 (0.85) DRD2DRD3ALDH1A1HTR1AHTR2A
SCHEMBL9196530 0.82 DRD2 (0.85) DRD2DRD3HTR1AHTR2A
SCHEMBL61850 0.81 DRD2 (0.66) DRD2DRD3CYP1A2CYP3A4CYP2C9
SCHEMBL9841829 0.80 DRD2 (0.81) DRD2DRD3HTR1AHTR2A
SCHEMBL9197525 0.80 DRD2 (0.81) DRD2DRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed