SCHEMBL9200735

SCHEMBL9200735

CCOC(=O)c1ccc(OCCCN2CCNCC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.72
KCNH2 Q12809 1/20 0.72
HRH2 P25021 12/20 0.67
HRH1 P35367 12/20 0.67
MEN1 O00255 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
KMT2A Q03164 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
TBXAS1 P24557 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199244 0.94 KCNH2 (0.63) HRH3KCNH2HRH2HRH1ALDH1A1
SCHEMBL4224568 0.87 HRH3 (0.93) HRH3KCNH2HRH2HRH1ALDH1A1
SCHEMBL5214308 0.85 HRH3 (0.72) HRH3KCNH2HRH2HRH1ALDH1A1
SCHEMBL7250762 0.84 KDM4E (0.70) HRH3HRH2HRH1MEN1ALDH1A1
SCHEMBL4096430 0.84 HRH3 (1.00) HRH3KCNH2HRH2HRH1ALDH1A1
SCHEMBL10899499 0.84 KCNH2 (0.57) HRH3KCNH2HRH2HRH1
Hydrochloric Acid SCHEMBL10900765 0.82 KCNH2 (0.56) HRH3KCNH2HRH2HRH1
SCHEMBL21408538 0.82 HRH3 (0.79) HRH3KCNH2HRH2HRH1MEN1
SCHEMBL13765617 0.81 HRH2 (0.59) HRH3KCNH2HRH2HRH1MEN1
SCHEMBL13044318 0.81 HRH2 (0.59) HRH3KCNH2HRH2HRH1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1037268-C Antipicornaviral pyridazinamines JANSSEM PHARMACEUTICA N V (BE) 1998-02-04 CN disclosed
EP-0435381-B1 Antipicornaviral pyridazinamines JANSSEN PHARMACEUTICA NV (BE) 1995-11-02 EP disclosed
EP-0398425-B1 Antirhinoviral piperidinyl, pyrrolidinyl and piperazinyl alkylphenol ethers JANSSEN PHARMACEUTICA NV (BE) 1994-03-16 EP disclosed
US-5196535-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-23 US disclosed
US-5100893-A Viricides, effective against picorna virus, durability JANSSEN PHARMACEUTICA N.V. (BE) 1992-03-31 US disclosed
EP-0435381-A1 Antipicornaviral pyridazinamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-07-03 EP disclosed
EP-0398425-A1 Antirhinoviral piperidinyl, pyrrolidinyl and piperazinyl alkylphenol ethers JANSSEN PHARMACEUTICA N.V. (BE) 1990-11-22 EP disclosed