SCHEMBL9200874

SCHEMBL9200874

OC1(c2cccnc2)CCC(N2CCN(c3ccccn3)CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
GRIN2B Q13224 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
HTR1A P08908 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9200867 1.00 ALDH1A1 (0.46) ALDH1A1LMNAGRIN2BHRH3HTR1A
SCHEMBL9200871 1.00 ALDH1A1 (0.46) ALDH1A1LMNAGRIN2BHRH3HTR1A
SCHEMBL9199399 0.90 GRIN2B (0.55) GRIN2BHRH3HTR1AADRA1DADRA1A
SCHEMBL9841972 0.84 DRD2 (0.43) DRD2
SCHEMBL9196215 0.84 CCR1 (0.48) ALDH1A1
SCHEMBL9842132 0.84 CCR1 (0.48) ALDH1A1
SCHEMBL9196219 0.84 CCR1 (0.48) ALDH1A1
SCHEMBL9196218 0.84 CCR1 (0.48) ALDH1A1
SCHEMBL9202976 0.83 HRH3 (0.48) HRH3HTR1AADRA1DADRA1AADRA1B
SCHEMBL9202985 0.83 HRH3 (0.48) HRH3HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4975445-A Antidepressants WARNER-LAMBERT COMPANY (US) 1990-12-04 US disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed