SCHEMBL9201072

SCHEMBL9201072

c1cnc2c(c1)C1(c3cccnc3-2)C(c2cnccn2)CCCC1c1cnccn1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.35
PDK2 Q15119 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
NPY5R Q15761 1/20 0.32
GSK3B P49841 1/20 0.32
CYP11B2 P19099 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9195303 0.83 CYP2A6 (0.36) CYP2A6PDK2CYP1A2CYP2C19KMT2A
SCHEMBL9545132 0.81 CYP11B2 (0.45) CYP2A6CYP1A2CYP2C19KMT2ACYP11B2
SCHEMBL9545168 0.79 PDK2 (0.35) PDK2CYP1A2CYP2C19KMT2A
SCHEMBL9275393 0.78 PDK2 (0.33) PDK2CYP1A2CYP2C19KMT2ACYP11B2
SCHEMBL9545528 0.71 GSK3B (0.38) PDK2CYP1A2CYP2C19KMT2AGSK3B
SCHEMBL9194471 0.70 GSK3B (0.47) PDK2CYP1A2CYP2C19KMT2AGSK3B
SCHEMBL9200820 0.68 CYP2A6 (0.40) CYP2A6CYP1A2CYP2C19KMT2ACYP11B2
SCHEMBL9545525 0.66 PDK2 (0.32) PDK2CYP1A2CYP2C19KMT2A
SCHEMBL28197535 0.65 MAP4K4 (0.40) NPY5RCYP11B2
SCHEMBL9198802 0.65 NFKB1 (0.45) PDK2CYP1A2CYP2C19KMT2ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636132-A1 SUBSTITUTED NITROGEN CONTAINING SPIRO COMPOUNDS FOR USE IN TREATING COGNITIVE DEFICITS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-02-01 EP disclosed