SCHEMBL9201400

SCHEMBL9201400

CCCC[CH]c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 6/20 0.44
HTR7 P34969 1/20 0.41
NFE2L2 Q16236 3/20 0.40
KMT2A Q03164 2/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
LMNA P02545 2/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PSMD14 O00487 1/20 0.37
HSP90AA1 P07900 1/20 0.37
MMP2 P08253 1/20 0.37
MC4R P32245 1/20 0.37
RAD52 P43351 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5878874 0.94 TRPA1 (0.42) TRPA1HTR7NFE2L2KMT2AHPGD
SCHEMBL6320373 0.89 ALDH1A1 (0.39) KMT2AHPGDLMNAMAPTNPSR1
SCHEMBL653095 0.86 NFE2L2 (0.43) TRPA1NFE2L2KMT2ALMNAMEN1
SCHEMBL1612718 0.80 CYP2A6 (0.46) NFE2L2HPGDL3MBTL1MAPTNPSR1
SCHEMBL15050819 0.79 NFE2L2 (0.47) TRPA1HTR7NFE2L2PTGS1PTGS2
SCHEMBL15050816 0.79 NFE2L2 (0.47) TRPA1HTR7NFE2L2PTGS1PTGS2
SCHEMBL654529 0.79 NFE2L2 (0.48) TRPA1NFE2L2KMT2ALMNAMEN1
SCHEMBL1611354 0.78 ALDH1A1 (0.46) KMT2AHPGDL3MBTL1PTGS1PTGS2
SCHEMBL27916482 0.78 LMNA (0.44) KMT2AHPGDL3MBTL1LMNAMEN1
SCHEMBL6422361 0.78 ALDH1A1 (0.47) KMT2APTGS1PTGS2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0650476-A1 PERIPHERAL VASODILATING AGENT CONTAINING N-ACYLATED 4-AMINO PIPERIDINE DERIVATIVES AS ACTIVE INGREDIENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-03 EP disclosed
WO-1994022826-A1 PERIPHERAL VASODILATING AGENT CONTAINING N-ACYLATED 4-AMINO PIPERIDINE DERIVATIVES AS ACTIVE INGREDIENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-13 WO disclosed