SCHEMBL9201461

SCHEMBL9201461

C1=CC=CN(Cc2ccccc2)C=C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.46
ELANE P08246 2/20 0.44
F2 P00734 1/20 0.44
PLG P00747 1/20 0.44
CTSG P08311 1/20 0.44
CMA1 P23946 1/20 0.44
CTRC Q99895 1/20 0.44
CYP19A1 P11511 2/20 0.43
GSK3A P49840 2/20 0.41
GSK3B P49841 2/20 0.41
MGLL Q99685 1/20 0.41
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
CALM1 P0DP23 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8672368 0.89 SIGMAR1 (0.41) SIGMAR1ELANEF2PLGCTSG
SCHEMBL24938710 0.78 MGLL (0.45) SIGMAR1ELANEF2PLGCTSG
SCHEMBL27675286 0.78 S1PR5 (0.47) LMNASMN1; SMN2KDM4EMEN1ALDH1A1
SCHEMBL30445901 0.78 CYP19A1 (0.38) SIGMAR1ELANEF2PLGCTSG
SCHEMBL6705444 0.76 SIGMAR1 (0.48) SIGMAR1ELANEF2PLGCTSG
Hydrochloric Acid SCHEMBL28835985 0.76 MGLL (0.43) SIGMAR1ELANEF2PLGCTSG
SCHEMBL21104726 0.76 SIGMAR1 (0.43) SIGMAR1ELANEF2PLGCTSG
SCHEMBL6615669 0.76 GSK3A (0.36) SIGMAR1ELANEF2PLGCTSG
Hydrochloric Acid SCHEMBL30234811 0.75 MGLL (0.42) SIGMAR1ELANEF2PLGCTSG
SCHEMBL27706105 0.75 SIGMAR1 (0.41) SIGMAR1ELANEF2PLGCTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107879967-A The preparation method of the ketone of 1 azaspiro [4.4] nonane 6 上海交通大学 2018-04-06 CN claimed
CN-104470547-B Utilize the method for tubular article synthesis of radiopharmaceuticals 未来化学株式会社 2018-01-26 CN claimed
CN-106459011-B Sigma-2 receptor ligand drug conjugates as antitumor compounds, methods of synthesis thereof and uses thereof 华盛顿大学 2019-11-15 CN disclosed
CN-109796482-A The preparation method of di-oxalate lithium borate and LiBF4 江苏长园华盛新能源材料有限公司 2019-05-24 CN disclosed
CN-105085515-B Hydrazide kind compound as coagulation factor xa inhibitors 华北制药股份有限公司 2019-02-01 CN disclosed
CN-107879967-A The preparation method of the ketone of 1 azaspiro [4.4] nonane 6 上海交通大学 2018-04-06 CN disclosed
CN-106459011-A Sigma-2 receptor ligand drug conjugates as antitumor compounds, methods of synthesis thereof and uses thereof 华盛顿大学 2017-02-22 CN disclosed
CN-103562181-A Method for producing hemiaminal compound and method for producing cyanoamine compound SUMITOMO CHEMICAL CO 2014-02-05 CN disclosed
CN-102356082-A 3,3' -spiroindolinone derivatives as anticancer agents HOFFMANN LA ROCHE 2012-02-15 CN disclosed
CN-101715452-A Azaindole-indole coupled derivatives, preparation methods and uses thereof JINGCAI CHENG 2010-05-26 CN disclosed
CN-101208085-A Modified release formulations of 1- [ (3-hydroxy-adamantyl-1-ylamino) -acetyl ] -pyrrolidinyl-2(s) -carbonitrile NOVARTIS AG (CH) 2008-06-25 CN disclosed
EP-0687249-A1 BALANOIDS ELI LILLY AND COMPANY (US) 1995-12-20 EP disclosed
WO-1994020062-A2 BALANOIDS AS PROTEIN KINASE C INHIBITORS ELI LILLY AND COMPANY (US) 1994-09-15 WO disclosed
CN-86106702-A The preparation method of azepine-3-cyclobutane-carboxylic acid and salt thereof 1987-04-01 CN disclosed