SCHEMBL9201720

SCHEMBL9201720

Cc1nc(-c2cc(C)c(OCCCCCc3cc(CO)no3)c(C)c2)no1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
NR1I2 O75469 1/20 0.52
PPARA Q07869 1/20 0.35
S1PR1 P21453 8/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK14 Q16539 2/20 0.34
S1PR3 Q99500 4/20 0.33
SCARB1 Q8WTV0 1/20 0.33
HTR1D P28221 4/20 0.32
HTR1B P28222 4/20 0.32
HTR2A P28223 4/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9520549 0.88 CYP3A4 (0.51) CYP3A4CYP2D6NR1I2PPARAS1PR1
SCHEMBL9521817 0.88 CYP3A4 (0.51) CYP3A4CYP2D6NR1I2PPARAS1PR1
SCHEMBL9202945 0.86 NR1I2 (0.67) CYP3A4CYP2D6NR1I2S1PR1L3MBTL1
SCHEMBL9205929 0.85 NR1I2 (0.57) CYP3A4CYP2D6NR1I2S1PR1L3MBTL1
SCHEMBL9203587 0.84 NR1I2 (0.56) CYP3A4CYP2D6NR1I2PPARAS1PR1
SCHEMBL9521718 0.83 CYP3A4 (0.55) CYP3A4CYP2D6NR1I2S1PR1L3MBTL1
SCHEMBL9207040 0.83 NR1I2 (0.44) CYP3A4CYP2D6NR1I2PPARAS1PR1
SCHEMBL8135581 0.82 CYP3A4 (0.52) CYP3A4CYP2D6NR1I2S1PR1L3MBTL1
SCHEMBL5099352 0.82 NR1I2 (0.77) CYP3A4CYP2D6NR1I2
SCHEMBL9201818 0.82 NR1I2 (0.39) CYP3A4CYP2D6NR1I2PPARAS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0413289-B1 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC (US) 1995-02-01 EP disclosed
US-5175178-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING DRUG INC. (US) 1992-12-29 US disclosed
US-4942241-A PICORNAVIRUS INCLUDING RHINOVIRUS STERLING DRUG INC. (US) 1990-07-17 US disclosed