SCHEMBL9201765

SCHEMBL9201765

COC(=O)c1cnn(C)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
KMT2A Q03164 3/20 0.42
TSHR P16473 2/20 0.41
LMNA P02545 1/20 0.41
NR4A2 P43354 1/20 0.41
BRD4 O60885 1/20 0.40
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 3/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39
CYP2C9 P11712 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9204354 0.82 CYP1A2 (0.44) CYP1A2CYP2C19KMT2ATSHRNR4A2
SCHEMBL28965242 0.81 CYP1A2 (0.50) CYP1A2CYP2C19KMT2ATSHRNR4A2
SCHEMBL10184712 0.81 KMT2A (0.53) CYP1A2CYP2C19KMT2ATSHRLMNA
SCHEMBL4701434 0.80 RAB9A (0.49) KMT2ATSHRLMNAKDM4EALDH1A1
SCHEMBL27941481 0.79 SMN1; SMN2 (0.38) LMNAKDM4EALDH1A1NPC1HPGD
SCHEMBL9196622 0.79 CYP1A2 (0.43) CYP1A2CYP2C19KMT2ATSHRLMNA
SCHEMBL26654708 0.79 CYP1A2 (0.49) CYP1A2CYP2C19KMT2ATSHRLMNA
SCHEMBL17895911 0.79 CYP1A2 (0.46) CYP1A2CYP2C19KMT2ATSHRLMNA
SCHEMBL3436120 0.79 CYP1A2 (0.51) CYP1A2CYP2C19KMT2ATSHRLMNA
SCHEMBL9105724 0.78 CYP1A2 (0.48) CYP1A2CYP2C19KMT2ATSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181150-A Pyrazole amide derivative, preparation method and application thereof 沈阳万菱生物技术有限公司 2022-03-15 CN claimed
CN-114181150-A Pyrazole amide derivative, preparation method and application thereof 沈阳万菱生物技术有限公司 2022-03-15 CN disclosed
EP-0087780-B2 Pyrazolesulfonylurea derivative, preparation thereof, herbicide containing said derivative as active ingredient and herbicidal method by use thereof NISSAN CHEMICAL IND LTD (JP) 1995-02-15 EP disclosed
US-4954164-A Pyrazolesulfonylurea derivatives, preparation thereof, herbicide containing said derivative as active ingredient and herbicidal method by use thereof NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-04 US disclosed