SCHEMBL9202912

SCHEMBL9202912

OC1(c2ccccn2)CCC(CCN2C=CC(C3=CCC=CC3)=CC2)CC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9200945 0.84 MEN1 (0.34) CCR1OPRM1OPRL1HSD11B1
SCHEMBL9204637 0.82 OPRM1 (0.35) CCR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL9773141 0.74 DRD2 (0.31)
SCHEMBL9201872 0.72
SCHEMBL9200022 0.68 DRD2 (0.60) CCR1
SCHEMBL9202901 0.68 DRD2 (0.60) CCR1
SCHEMBL9200032 0.68 DRD2 (0.60) CCR1
SCHEMBL9196526 0.67 DRD2 (0.59)
SCHEMBL9467917 0.66
SCHEMBL30790731 0.65 OPRM1 (0.48) CCR1OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed