SCHEMBL9200945

SCHEMBL9200945

OC1(c2cccnc2)CCC(CCN2C=CC(C3=CCC=CC3)=CC2)CC1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CCR1 P32246 1/20 0.34
ALDH1A1 P00352 6/20 0.33
PKM P14618 1/20 0.33
LMNA P02545 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRL1 P41146 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
AR P10275 1/20 0.32
KCNH2 Q12809 1/20 0.32
GAA P10253 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
HSD11B1 P28845 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9202912 0.84 CCR1 (0.33) CCR1OPRM1OPRL1HSD11B1
SCHEMBL9199083 0.82 OPRM1 (0.37) MEN1KMT2AALDH1A1PKMLMNA
SCHEMBL9773141 0.74 DRD2 (0.31)
SCHEMBL9201872 0.72
SCHEMBL8906856 0.71 DRD2 (0.46)
SCHEMBL9379229 0.70 DRD2 (0.37)
SCHEMBL8908126 0.70 DRD2 (0.42)
Hydrochloric Acid SCHEMBL7783716 0.70 DRD2 (0.36)
SCHEMBL9373797 0.68 CHRNB2 (0.31)
SCHEMBL9200941 0.67 DRD2 (0.54) MEN1KMT2ACCR1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed