SCHEMBL9203045

SCHEMBL9203045

N[C@H]1CC[C@H](N2CCN(c3ccccn3)CC2)CC1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.56
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
ADRA1B P35368 1/20 0.56
HRH3 Q9Y5N1 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201106 1.00 HTR1A (0.56) HTR1AADRA1DADRA1AADRA1BHRH3
SCHEMBL3879984 1.00 HTR1A (0.56) HTR1AADRA1DADRA1AADRA1BHRH3
SCHEMBL28161959 0.84 HRH3 (0.60) HTR1AADRA1DADRA1AADRA1BHRH3
SCHEMBL29683564 0.84 PLD1 (0.58) HRH3
SCHEMBL243658 0.84 PLD1 (0.58) HRH3
SCHEMBL19823057 0.82 HTR1A (0.70) HTR1AADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL17557596 0.82 PLD1 (0.56) HRH3
Hydrochloric Acid SCHEMBL243428 0.82 PLD1 (0.56) HRH3
SCHEMBL3882641 0.82 HTR1A (0.51) HTR1AADRA1DADRA1AADRA1BHRH3
SCHEMBL7898534 0.81 DRD2 (0.44) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed