SCHEMBL9203671

SCHEMBL9203671

COC(=O)COc1cc(OCC=Cc2ccccc2)cc(OCC(=O)OC)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
RAB9A P51151 2/20 0.53
PTGS2 P35354 2/20 0.51
CYSLTR2 Q9NS75 1/20 0.50
CYSLTR1 Q9Y271 1/20 0.50
KMT2A Q03164 3/20 0.48
LTB4R Q15722 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.47
PPARA Q07869 3/20 0.47
PPARD Q03181 2/20 0.47
PPARG P37231 2/20 0.47
MEN1 O00255 2/20 0.47
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9203661 1.00 NPC1 (0.53) NPC1RAB9APTGS2CYSLTR2CYSLTR1
SCHEMBL9206284 0.93 LTB4R (0.53) NPC1RAB9APTGS2CYSLTR2CYSLTR1
SCHEMBL9206279 0.93 LTB4R (0.53) NPC1RAB9APTGS2CYSLTR2CYSLTR1
SCHEMBL9201444 0.85 LTB4R (0.54) NPC1RAB9AKMT2ALTB4RLTB4R2
SCHEMBL9201451 0.85 LTB4R (0.54) NPC1RAB9AKMT2ALTB4RLTB4R2
SCHEMBL9199980 0.85 LTB4R (0.66) NPC1RAB9ACYSLTR2CYSLTR1KMT2A
SCHEMBL9206318 0.84 LTB4R (0.59) NPC1RAB9AKMT2ALTB4RLTB4R2
SCHEMBL9206314 0.84 LTB4R (0.59) NPC1RAB9AKMT2ALTB4RLTB4R2
SCHEMBL9201817 0.82 LTB4R (0.77) LTB4RLTB4R2
SCHEMBL9857423 0.81 IDO1 (0.47) NPC1RAB9APTGS2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538416-B1 SUBSTITUTED MONOCYCLIC ARYL COMPOUNDS EXHIBITING SELECTIVE LEUKOTRIENE B 4 ANTAGONIST ACTIVITY RHONE POULENC RORER INT (US) 1995-08-09 EP disclosed
US-5232948-A SUBSTITUTED MONOCYCLIC ARYL COMPOUNDS EXHIBITING SELECTIVE LEUKOTRIENE B4 ANTAGONIST ACTIVITY RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1993-08-03 US disclosed