SCHEMBL9205301

SCHEMBL9205301

O=C(O)CN1CCN(CC(=O)O)Cc2cccc(n2)C1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.40
SLC6A9 P48067 1/20 0.40
POLB P06746 1/20 0.40
PDE4B Q07343 1/20 0.38
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
HSD17B10 Q99714 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
AKR1B1 P15121 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
KMT2A Q03164 1/20 0.37
TGM2 P21980 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1394889 0.98 SLC6A9 (0.42) EGLN1SLC6A9POLBPDE4BALDH1A1
SCHEMBL20624199 0.94 EGLN1 (0.36) EGLN1SLC6A9POLBPDE4BKDM4E
SCHEMBL7869921 0.94 EGLN1 (0.39) EGLN1SLC6A9POLBPDE4BALDH1A1
SCHEMBL12544369 0.92 CYP2C19 (0.43) ALDH1A1KDM4EMEN1KMT2A
SCHEMBL7871400 0.92 ALDH1A1 (0.40) EGLN1POLBALDH1A1KDM4EMEN1
SCHEMBL16800534 0.91 NOS1 (0.43) EGLN1SLC6A9PDE4BALDH1A1GAA
SCHEMBL29299528 0.91 NOS1 (0.43) EGLN1SLC6A9PDE4BALDH1A1GAA
SCHEMBL22887713 0.90 SLC6A9 (0.41) EGLN1SLC6A9POLBPDE4BALDH1A1
SCHEMBL12747963 0.89 CYP2C19 (0.41) PDE4BALDH1A1GAAKDM4EMEN1
SCHEMBL25574097 0.89 ALDH1A1 (0.45) EGLN1SLC6A9ALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
EP-0352218-B1 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AG (DE) 1995-02-22 EP disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0352218-A2 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-24 EP disclosed