SCHEMBL9205462

SCHEMBL9205462

Cc1cc2c(cc1C)C(=O)N(CC1CCCN(CCCc3c[nH]c4ccccc34)C1)CC2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.45
DRD2 P14416 2/20 0.44
HTR2A P28223 2/20 0.44
SLC6A4 P31645 1/20 0.44
HTR7 P34969 1/20 0.44
HRH1 P35367 1/20 0.44
DRD3 P35462 1/20 0.44
MAPT P10636 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GRM5 P41594 1/20 0.40
BCHE P06276 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9215340 0.95 HTR1A (0.47) HTR1ADRD2HTR2ASLC6A4HTR7
Hydrochloric Acid SCHEMBL9212006 0.94 HTR1A (0.46) HTR1ADRD2HTR2ASLC6A4HTR7
Water SCHEMBL9208576 0.93 HTR1A (0.39) HTR1ADRD2HTR2ASLC6A4HTR7
SCHEMBL9216130 0.85 HTR1A (0.47) HTR1ADRD2HTR2ASLC6A4HTR7
Hydrochloric Acid SCHEMBL10649448 0.83 HTR1A (0.54) HTR1ADRD2HTR2ASLC6A4HTR7
SCHEMBL9740802 0.83 SIGMAR1 (0.45) GRM5BCHE
Hydrochloric Acid SCHEMBL9205345 0.83 HTR1A (0.53) HTR1ADRD2HTR2ASLC6A4HTR7
SCHEMBL9215429 0.83 HTR1A (0.47) HTR1ADRD2HTR2ASLC6A4HTR7
Hydrochloric Acid SCHEMBL9741187 0.81 PDE4D (0.48) HTR1ADRD2HTR2ASLC6A4HTR7
SCHEMBL9207074 0.80 GRM5 (0.42) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed