SCHEMBL9205705

SCHEMBL9205705

COc1cccnc1N1CCN(CCCc2c[nH]c3ccc(F)cc23)CC1

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.73
SLC6A4 P31645 5/20 0.73
HTR7 P34969 4/20 0.73
KCNH2 Q12809 4/20 0.73
MPO P05164 3/20 0.63
SLC6A2 P23975 1/20 0.60
SLC6A3 Q01959 1/20 0.60
HTR6 P50406 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214152 0.94 HTR1A (0.65) HTR1ASLC6A4HTR7KCNH2MPO
SCHEMBL9210187 0.89 HTR1A (0.64) HTR1ASLC6A4HTR7KCNH2HTR6
SCHEMBL4357142 0.87 HTR1A (0.68) HTR1ASLC6A4HTR7KCNH2MPO
Hydrochloric Acid SCHEMBL9206187 0.87 HTR1A (0.62) HTR1ASLC6A4HTR7KCNH2HTR6
Hydrochloric Acid SCHEMBL4347864 0.86 HTR1A (0.70) HTR1ASLC6A4HTR7KCNH2MPO
Hydrochloric Acid SCHEMBL4356376 0.86 HTR1A (0.70) HTR1ASLC6A4HTR7KCNH2MPO
SCHEMBL9210900 0.86 HTR1A (0.65) HTR1ASLC6A4HTR7KCNH2HTR6
SCHEMBL27989611 0.85 HTR1A (0.69) HTR1AKCNH2HTR6
SCHEMBL9211546 0.85 HTR2A (0.64) HTR1A
Hydrochloric Acid SCHEMBL9213478 0.85 HTR1A (0.64) HTR1ASLC6A4HTR7KCNH2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP claimed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US claimed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP claimed