SCHEMBL9214152

SCHEMBL9214152

COc1cccnc1N1CCN(CCc2c[nH]c3ccc(F)cc23)CC1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 12/20 0.65
HTR7 P34969 7/20 0.65
KCNH2 Q12809 3/20 0.65
SLC6A4 P31645 3/20 0.65
MPO P05164 4/20 0.62
HTR6 P50406 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9205705 0.94 HTR1A (0.73) HTR1AHTR7KCNH2SLC6A4MPO
SCHEMBL9211546 0.90 HTR2A (0.64) HTR1A
SCHEMBL9213895 0.90 KCNH2 (0.59) HTR1AHTR7KCNH2SLC6A4MPO
SCHEMBL9205321 0.89 DRD2 (0.52) HTR1AHTR7KCNH2SLC6A4MPO
SCHEMBL9205349 0.88 ABCC1 (0.57) HTR1AHTR7KCNH2SLC6A4HTR6
SCHEMBL6362404 0.87 HTR1A (0.60) HTR1AHTR7KCNH2SLC6A4MPO
SCHEMBL9274974 0.85 DRD2 (0.57) HTR1A
SCHEMBL9210187 0.82 HTR1A (0.64) HTR1AHTR7KCNH2SLC6A4HTR6
SCHEMBL9210900 0.82 HTR1A (0.65) HTR1AHTR7KCNH2SLC6A4HTR6
SCHEMBL4357142 0.81 HTR1A (0.68) HTR1AHTR7KCNH2SLC6A4MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP claimed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US claimed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP claimed