SCHEMBL9211546

SCHEMBL9211546

COc1ccc2[nH]cc(CCN3CCN(c4ncccc4OC)CC3)c2c1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.64
HTR1A P08908 9/20 0.61
DRD2 P14416 2/20 0.58
ADRA2A P08913 1/20 0.58
ADRA2B P18089 1/20 0.58
ADRA2C P18825 1/20 0.58
ADRA1D P25100 1/20 0.58
ADRA1A P35348 1/20 0.58
ADRA1B P35368 1/20 0.58
DRD4 P21917 1/20 0.57
DRD3 P35462 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9274974 0.92 DRD2 (0.57) HTR2AHTR1ADRD2ADRA2AADRA2B
SCHEMBL9214152 0.90 HTR1A (0.65) HTR1A
SCHEMBL9213895 0.90 KCNH2 (0.59) HTR2AHTR1ADRD2DRD4DRD3
SCHEMBL9205321 0.89 DRD2 (0.52) HTR2AHTR1ADRD2DRD4DRD3
SCHEMBL9205349 0.88 ABCC1 (0.57) HTR2AHTR1ADRD2DRD4DRD3
SCHEMBL9205705 0.85 HTR1A (0.73) HTR1A
SCHEMBL9210187 0.82 HTR1A (0.64) HTR2AHTR1ADRD2ADRA1DADRA1A
SCHEMBL9210900 0.82 HTR1A (0.65) HTR2AHTR1ADRD2DRD4DRD3
SCHEMBL27989611 0.81 HTR1A (0.69) HTR1A
Hydrochloric Acid SCHEMBL9206187 0.81 HTR1A (0.62) HTR2AHTR1ADRD2ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP claimed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US claimed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP claimed