SCHEMBL9206013

SCHEMBL9206013

c1ccc2c3c([nH]c2c1)CCNC3CN1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 2/20 0.43
DRD2 P14416 2/20 0.43
DRD5 P21918 1/20 0.42
GRIN2B Q13224 1/20 0.41
CASP1 P29466 1/20 0.41
HTR2A P28223 3/20 0.40
HTR2C P28335 3/20 0.40
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866845 0.99 DRD1 (0.42) DRD1DRD2DRD5GRIN2BCASP1
SCHEMBL30149565 0.76 HTR2A (0.51) DRD2GRIN2BHTR2AHTR2CDRD3
SCHEMBL9865550 0.76 MEN1 (0.43) DRD1DRD2GRIN2BHTR2AHTR2C
Hydrochloric Acid SCHEMBL30149473 0.75 HTR2A (0.53) GRIN2BHTR2AHTR2CSIGMAR1
SCHEMBL9865545 0.75 MEN1 (0.42) DRD1DRD2GRIN2BHTR2AHTR2C
SCHEMBL14863014 0.70 MAPKAPK2 (0.62) DRD1DRD2HTR2AHTR2CSIGMAR1
SCHEMBL3453173 0.70 OPRM1 (0.56)
SCHEMBL329828 0.69 OPRM1 (0.57)
SCHEMBL329925 0.69 OPRM1 (0.57)
SCHEMBL31020939 0.69 HTR2A (0.44) DRD1DRD2GRIN2BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0333427-B1 Heterocyclic derivatives SMITHKLINE BEECHAM FARMA (IT) 1995-08-23 EP claimed
US-4999359-A Analgesics DR. LO ZAMBELETTI S.P.A. (IT) 1991-03-12 US disclosed