SCHEMBL9206944

SCHEMBL9206944

NC(=O)c1c(C2CCc3ccccc32)ccc2c1OCO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
MGAM O43451 1/20 0.36
AMY1A P0DUB6 1/20 0.36
GAA P10253 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
DRD2 P14416 3/20 0.36
HTR2A P28223 3/20 0.36
DRD3 P35462 3/20 0.36
PARP1 P09874 1/20 0.36
FABP4 P15090 1/20 0.36
MCHR1 Q99705 1/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
NTRK1 P04629 3/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3460627 0.71 PIN1 (0.49) TAS1R3TAS1R1PARP1CA1CA2
SCHEMBL3462221 0.71 PIN1 (0.49) TAS1R3TAS1R1PARP1CA1CA2
SCHEMBL2798590 0.71 PIN1 (0.49) TAS1R3TAS1R1PARP1CA1CA2
SCHEMBL422232 0.67 AOC3 (0.47) ALDH1A1
SCHEMBL18249682 0.65 ADRA1A (0.37) ALDH1A1TAS1R3TAS1R1FABP4MCHR1
SCHEMBL8516606 0.65 PIN1 (0.46) PARP1AURKARPS6KB1
SCHEMBL9814122 0.64 KCNH2 (0.39) ALDH1A1MGAMAMY1AGAASI
SCHEMBL27552078 0.64 TAS1R3 (0.40) TAS1R3TAS1R1
SCHEMBL28195960 0.64 ADRA1A (0.42) TAS1R3TAS1R1CA1CA2HSD11B1
SCHEMBL4276692 0.64 PIN1 (0.42) TAS1R3TAS1R1PARP1HSD11B1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612244-A4 ENDOTHELIN RECEPTOR ANTAGONISTS. SMITHKLINE BEECHAM CORP (US) 1995-05-17 EP disclosed
EP-0612244-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-08-31 EP disclosed