SCHEMBL9207748

SCHEMBL9207748

CCOC(=O)CN1CCN(CC(=O)OCC)Cc2ccc(o2)CN(CC(=O)OCC)CC1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
GSK3B P49841 2/20 0.41
GSK3A P49840 1/20 0.41
ALDH1A1 P00352 2/20 0.41
PIN1 Q13526 1/20 0.41
PIN4 Q9Y237 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
RAB9A P51151 1/20 0.41
HTR1A P08908 1/20 0.40
HTR2C P28335 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
ALOX15 P16050 1/20 0.38
GAA P10253 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11852921 0.80
SCHEMBL8912811 0.80 MGAM (0.50) KDM4EGSK3BGSK3AALDH1A1PIN1
SCHEMBL2373233 0.80 MGAM (0.50) KDM4EGSK3BGSK3AALDH1A1PIN1
SCHEMBL3966571 0.80 MGAM (0.50) KDM4EGSK3BGSK3AALDH1A1PIN1
SCHEMBL9213081 0.77 HSD17B10 (0.46) ALDH1A1SMN1; SMN2HSD17B10ITGB3ITGA2B
SCHEMBL8260387 0.75 MEN1 (0.47) KDM4EGSK3BGSK3AALDH1A1MEN1
SCHEMBL29419289 0.75 ALDH1A1 (0.45) KDM4EGSK3BGSK3AALDH1A1MEN1
SCHEMBL689078 0.75 LMNA (0.45) KDM4EGSK3BGSK3AALDH1A1PIN1
SCHEMBL8911750 0.73 HSD17B10 (0.44) KDM4EGSK3BGSK3AALDH1A1PIN1
SCHEMBL15997367 0.73 HSD17B10 (0.44) KDM4EGSK3BGSK3AALDH1A1PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
EP-0352218-B1 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AG (DE) 1995-02-22 EP disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0352218-A2 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-24 EP disclosed