SCHEMBL9207882

SCHEMBL9207882

Nc1cccc(OCCCNCC2COc3ccccc3O2)c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA4 P22748 1/20 0.59
CA5A P35218 1/20 0.59
CA9 Q16790 1/20 0.59
CA5B Q9Y2D0 1/20 0.59
ADRA1D P25100 6/20 0.57
ADRA1A P35348 6/20 0.57
ADRA1B P35368 6/20 0.57
HTR1A P08908 4/20 0.57
ALDH1A1 P00352 3/20 0.57
MEN1 O00255 2/20 0.57
CYP3A4 P08684 2/20 0.57
KMT2A Q03164 2/20 0.57
KDM4E B2RXH2 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
TSHR P16473 1/20 0.57
MAPK1 P28482 1/20 0.57
CYP2C19 P33261 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214181 1.00 CA1 (0.59) CA1CA2CA4CA5ACA9
SCHEMBL9210885 0.89 ADRA1D (0.52) CA1CA2CA4CA5ACA9
SCHEMBL9206070 0.89 ADRA1D (0.52) CA1CA2CA4CA5ACA9
SCHEMBL9203733 0.89 ADRA1D (0.52) CA1CA2CA4CA5ACA9
SCHEMBL9205182 0.89 ADRA1D (0.52) CA1CA2CA4CA5ACA9
SCHEMBL9210884 0.89 DRD2 (0.53)
SCHEMBL9207245 0.89 ADRA1D (0.49) CA1CA2CA4CA5ACA9
SCHEMBL9205645 0.89 DRD2 (0.53)
SCHEMBL9207871 0.89 ADRA1D (0.49) CA1CA2CA4CA5ACA9
SCHEMBL9205633 0.89 DRD2 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5126366-A Antidepressants, antipsychotics, anxiolytic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-30 US claimed
EP-0520674-B1 Antipsychotic benzodioxan derivatives AMERICAN HOME PROD (US) 1995-08-16 EP disclosed
EP-0520674-A1 Antipsychotic benzodioxan derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1992-12-30 EP disclosed
US-5126366-A Antidepressants, antipsychotics, anxiolytic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-30 US disclosed