SCHEMBL9208423

SCHEMBL9208423

O=C(O)CN1CCN(CC(=O)O)CC2CCC(CN(CC(=O)O)CC1)O2

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.47
PIK3CD O00329 1/20 0.41
SLC6A9 P48067 1/20 0.35
ITGB3 P05106 5/20 0.33
ITGA2B P08514 5/20 0.33
KDM4E B2RXH2 1/20 0.32
ACE P12821 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32
S1PR1 P21453 1/20 0.31
FOLH1 Q04609 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29946293 0.90 PIK3CD (0.45) HSD17B10PIK3CDACE
Trifluoroacetic Acid SCHEMBL28956754 0.80 PIK3CD (0.38) HSD17B10PIK3CD
SCHEMBL29946381 0.79 HSD17B10 (0.43) HSD17B10PIK3CDKDM4E
SCHEMBL6848102 0.76 HSD17B10 (0.64) HSD17B10SLC6A9KDM4ES1PR1
Tetraxetan SCHEMBL18018 0.76 HSD17B10 (0.64) HSD17B10SLC6A9KDM4ES1PR1
Tetraxetan SCHEMBL2017956 0.76 HSD17B10 (0.64) HSD17B10SLC6A9KDM4ES1PR1
SCHEMBL321989 0.76 HSD17B10 (0.64) HSD17B10SLC6A9KDM4ES1PR1
SCHEMBL173508 0.76 HSD17B10 (0.64) HSD17B10SLC6A9KDM4ES1PR1
Tetraxetan SCHEMBL2635294 0.76 HSD17B10 (0.64) HSD17B10SLC6A9KDM4ES1PR1
SCHEMBL3660521 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
EP-0352218-B1 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AG (DE) 1995-02-22 EP disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0352218-A2 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-24 EP disclosed