SCHEMBL9208424

SCHEMBL9208424

CSc1ccc(-c2cc(CN)nn2-c2ccc(F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.49
PTGS1 P23219 5/20 0.49
KCNH2 Q12809 4/20 0.45
CHRNA7 P36544 1/20 0.42
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
CYP1A2 P05177 1/20 0.41
NR3C2 P08235 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ATM Q13315 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9203794 0.88 PTGS2 (0.48) PTGS2PTGS1KCNH2CHRNA7RXRA
SCHEMBL9205227 0.87 PTGS2 (0.51) PTGS2PTGS1KCNH2CHRNA7RXRA
SCHEMBL17378009 0.85 PTGS2 (0.54) PTGS2PTGS1KCNH2CHRNA7RXRA
SCHEMBL9211086 0.85 PTGS2 (0.45) PTGS2PTGS1KCNH2CHRNA7RXRA
SCHEMBL9202494 0.83 PTGS2 (0.52) PTGS2PTGS1CHRNA7MEN1KMT2A
SCHEMBL9207835 0.82 PTGS2 (0.51) PTGS2PTGS1CHRNA7MEN1KMT2A
SCHEMBL27742806 0.82 MEN1 (0.58) PTGS2PTGS1KCNH2RXRARXRB
SCHEMBL9208745 0.80 MALT1 (0.67) RXRARXRBRXRG
SCHEMBL9201624 0.80 PTGS2 (0.47) PTGS2PTGS1KCNH2CHRNA7RXRA
SCHEMBL9206412 0.80 PTGS2 (0.49) PTGS2PTGS1CHRNA7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed