SCHEMBL9209656

SCHEMBL9209656

COc1cc2c(cc1OC)CC(=O)N(CC1CCN(CCc3cccs3)C1)CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
TSHR P16473 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HCN4 Q9Y3Q4 2/20 0.42
MAPT P10636 1/20 0.42
CYP3A4 P08684 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 1/20 0.42
ATM Q13315 1/20 0.41
PKM P14618 1/20 0.41
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
SLC6A4 P31645 1/20 0.40
DRD3 P35462 1/20 0.40
KCNH2 Q12809 1/20 0.40
DRD1 P21728 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9741774 0.94 ALOX15 (0.45) ALOX15ALDH1A1KDM4ETSHRCASP1
SCHEMBL9215720 0.94 ALOX15 (0.45) ALOX15ALDH1A1KDM4ETSHRCASP1
SCHEMBL9216033 0.90 ATM (0.39) ALOX15ALDH1A1KDM4ETSHRCASP1
SCHEMBL9206630 0.89 ALOX15 (0.43) ALOX15ALDH1A1KDM4ETSHRCASP1
Hydrochloric Acid SCHEMBL9740340 0.88 ALOX15 (0.43) ALOX15ALDH1A1KDM4ETSHRCASP1
Hydrochloric Acid SCHEMBL9740263 0.88 ALOX15 (0.42) ALOX15ALDH1A1KDM4ETSHRCASP1
Hydrochloric Acid SCHEMBL9739549 0.88 ALOX15 (0.42) ALOX15ALDH1A1KDM4ETSHRCASP1
SCHEMBL9214406 0.86 ATM (0.37) ALDH1A1KDM4ESMN1; SMN2ATMDRD4
SCHEMBL9207422 0.85 HRH3 (0.40) ALOX15ALDH1A1KDM4ETSHRCASP1
SCHEMBL9208037 0.84 HRH3 (0.37) ALOX15ALDH1A1KDM4ETSHRCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed