SCHEMBL9216033

SCHEMBL9216033

Cc1cc2c(cc1C)CC(=O)N(CC1CCN(CCc3cccs3)C1)CC2

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.39
HRH3 Q9Y5N1 2/20 0.36
SHMT2 P34897 1/20 0.35
OPRM1 P35372 3/20 0.35
OPRD1 P41143 3/20 0.35
OPRK1 P41145 3/20 0.35
POLB P06746 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207422 0.94 HRH3 (0.40) ATMHRH3KDM4EALDH1A1ALOX15
SCHEMBL9208037 0.94 HRH3 (0.37) ATMHRH3POLBKDM4EALDH1A1
SCHEMBL9209656 0.90 ALOX15 (0.47) ATMKDM4EALDH1A1ALOX15TSHR
SCHEMBL9214406 0.89 ATM (0.37) ATMHRH3SHMT2OPRM1OPRD1
SCHEMBL9208876 0.88 HRH3 (0.36) HRH3KDM4EALDH1A1
SCHEMBL9212975 0.88 HRH3 (0.35) HRH3KDM4EALDH1A1
Hydrochloric Acid SCHEMBL9741774 0.84 ALOX15 (0.45) HRH3KDM4EALDH1A1ALOX15TSHR
SCHEMBL9215720 0.84 ALOX15 (0.45) ATMKDM4EALDH1A1ALOX15TSHR
SCHEMBL9207563 0.84 LTA4H (0.37) ATMHRH3OPRM1OPRD1OPRK1
SCHEMBL9205933 0.83 LTA4H (0.35) ATMHRH3OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed