SCHEMBL9209745

SCHEMBL9209745

CC(NCCOC(N)=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2D6 P10635 2/20 0.51
LMNA P02545 2/20 0.51
CASR P41180 2/20 0.51
CHRM2 P08172 1/20 0.51
HTR1A P08908 1/20 0.51
ADRA2A P08913 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
CHRM1 P11229 1/20 0.51
SMPD1 P17405 1/20 0.51
DRD1 P21728 1/20 0.51
TBXA2R P21731 1/20 0.51
SLC6A2 P23975 1/20 0.51
SLC6A4 P31645 1/20 0.51
ADRA1A P35348 1/20 0.51
OPRM1 P35372 1/20 0.51
DRD3 P35462 1/20 0.51
HTR2B P41595 1/20 0.51
SLC6A3 Q01959 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11400626 0.82 APAF1 (0.49) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL28945403 0.80 ALDH1A1 (0.44) LMNAKMT2AMEN1ALDH1A1
SCHEMBL8268348 0.76 LMNA (0.61) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL31248153 0.76 LMNA (0.61) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL28816657 0.76 CYP1A2 (0.54) CYP1A2CYP2D6LMNACHRM2CHRM1
SCHEMBL24406703 0.75 CYP3A4 (0.76) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL3881699 0.75 CYP3A4 (0.76) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL5471668 0.75 CYP3A4 (0.76) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL3881700 0.75 CYP3A4 (0.76) CYP1A2CYP3A4CYP2D6LMNACASR
SCHEMBL2432448 0.75 KCNH2 (0.50) CYP1A2CYP2D6LMNAHTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111943945-B Suvorexant intermediate and preparation method thereof 上海应用技术大学 2022-07-12 CN disclosed
CN-111943945-A Suvorexant intermediate and preparation method thereof 上海应用技术大学 2020-11-17 CN disclosed
EP-0655055-A1 TACHYKININ ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1995-05-31 EP disclosed