SCHEMBL9210258

SCHEMBL9210258

COc1cc2c(cc1OC)CC(=O)N(CC1CCCN(CCCCCc3cc4ccccc4o3)C1)CC2

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.44
HTR2B P41595 5/20 0.44
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 1/20 0.39
HCN4 Q9Y3Q4 1/20 0.39
CHRNB2 P17787 3/20 0.39
CHRNA4 P43681 3/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
ABCB1 P08183 3/20 0.39
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
DRD3 P35462 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210043 0.99 DRD2 (0.44) DRD2HTR2BHCRTR1HCRTR2SMN1; SMN2
SCHEMBL9207394 0.94 HCRTR1 (0.44) DRD2HTR2BHCRTR1HCRTR2SMN1; SMN2
SCHEMBL9210489 0.92 HCRTR1 (0.44) DRD2HTR2BHCRTR1HCRTR2SMN1; SMN2
SCHEMBL9206641 0.92 MAPK1 (0.41) DRD2HTR2BSMN1; SMN2CHRNB2CHRNA4
SCHEMBL9214809 0.91 MAPK1 (0.41) DRD2HTR2BHCRTR1HCRTR2SMN1; SMN2
SCHEMBL9216985 0.89 HTR2B (0.45) DRD2HTR2BHCRTR1HCRTR2SMN1; SMN2
SCHEMBL9209357 0.89 DRD2 (0.37) DRD2HTR2BSMN1; SMN2CHRNB2CHRNA4
SCHEMBL9208812 0.88 DRD2 (0.38) DRD2HTR2BSMN1; SMN2DRD3LMNA
SCHEMBL9215152 0.85 MAPK1 (0.44) DRD2HTR2BHCRTR1HCRTR2SMN1; SMN2
SCHEMBL9216928 0.83 HCRTR1 (0.41) HCRTR1HCRTR2SMN1; SMN2MAPTHCN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed