SCHEMBL9216928

SCHEMBL9216928

COc1cc2c(cc1OC)CC(=O)N(CC1CCCN(CCCc3cc4ccccc4s3)C1)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNB4 P30926 2/20 0.41
CHRNA3 P32297 2/20 0.41
CHRNA4 P43681 2/20 0.41
HCN4 Q9Y3Q4 2/20 0.40
MAPT P10636 1/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
CHRM2 P08172 1/20 0.38
HTR1A P08908 1/20 0.38
SLC6A4 P31645 1/20 0.38
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.38
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213551 0.95 HCRTR1 (0.42) HCRTR1HCRTR2CHRNB2CHRNB4CHRNA3
SCHEMBL9216368 0.91 KDM2B (0.36) HCRTR1HCRTR2KCNH2LMNAKDM2B
SCHEMBL9206763 0.88 LTA4H (0.36) HCRTR1HCRTR2LMNAKDM2B
SCHEMBL9215744 0.86 KDM2B (0.37) HCRTR1HCRTR2SLC6A4KCNH2LMNA
SCHEMBL9210043 0.84 DRD2 (0.44) HCRTR1HCRTR2CHRNB2CHRNB4CHRNA3
SCHEMBL9206630 0.83 ALOX15 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4HCN4
SCHEMBL9213547 0.83 LTA4H (0.37) HCRTR1HCRTR2LMNAKDM2B
SCHEMBL9210258 0.83 DRD2 (0.44) HCRTR1HCRTR2CHRNB2CHRNB4CHRNA3
SCHEMBL9207394 0.83 HCRTR1 (0.44) HCRTR1HCRTR2HCN4MAPTCYP3A4
Hydrochloric Acid SCHEMBL9740340 0.83 ALOX15 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4HCN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed