SCHEMBL9210338

SCHEMBL9210338

CC(=O)N1CCC(CCC(=O)c2ccc3c(c2)CCN3C(=O)C(F)(F)F)CC1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.52
ALDH1A1 P00352 6/20 0.49
HPGD P15428 3/20 0.49
KDM4E B2RXH2 3/20 0.47
RECQL P46063 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
MAPT P10636 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HSD17B10 Q99714 1/20 0.44
NOTUM Q6P988 1/20 0.44
MCHR1 Q99705 1/20 0.43
LMNA P02545 1/20 0.43
RAB9A P51151 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9205255 0.92 ACHE (0.49) ACHEALDH1A1MAPTMCHR1
SCHEMBL9208669 0.91 ALDH1A1 (0.59) ACHEALDH1A1HPGDKDM4ERECQL
SCHEMBL9210160 0.85 ACHE (0.69) ACHEALDH1A1HPGDMCHR1
SCHEMBL9208181 0.84 ACHE (0.57) ACHEALDH1A1HPGDKDM4ERECQL
SCHEMBL9212033 0.83 ACHE (0.54) ACHEALDH1A1HPGDKDM4ERECQL
SCHEMBL9208257 0.82 ACHE (0.70) ACHEALDH1A1HPGDMCHR1
SCHEMBL9208387 0.81 ACHE (0.70) ACHE
SCHEMBL7227822 0.80 MCHR1 (0.55) ACHEMCHR1
SCHEMBL7227474 0.78 ACHE (0.60) ACHEALDH1A1HPGDMCHR1
SCHEMBL9204837 0.78 ACHE (0.73) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487071-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-07-05 EP disclosed
US-5273974-A Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-28 US disclosed
EP-0487071-A1 Condensed heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-05-27 EP disclosed