SCHEMBL9210485

SCHEMBL9210485

CC1(N)CN(c2c(F)cc3c(=O)c(OC(=O)O)cn(CCF)c3c2Cl)C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.46
KCNH2 Q12809 2/20 0.40
ALDH1A1 P00352 5/20 0.38
POLB P06746 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TOP1 P11387 8/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
PMP22 Q01453 1/20 0.33
ADRA2B P18089 1/20 0.33
MAPK1 P28482 1/20 0.33
TOP2A P11388 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9668111 0.92 KDM4E (0.55) KDM4EKCNH2ALDH1A1TOP1HPGD
SCHEMBL9148013 0.88 KDM4E (0.60) KDM4EKCNH2ALDH1A1POLBCHRM2
SCHEMBL9215533 0.83 ALDH1A1 (0.54) KDM4EKCNH2ALDH1A1POLBCHRM2
SCHEMBL9668418 0.83 HSD17B10 (0.48) KDM4EKCNH2ALDH1A1CYP2C9HPGD
SCHEMBL9213820 0.83 CYP3A4 (0.39) KDM4EKCNH2ALDH1A1POLBCHRM2
SCHEMBL9217114 0.82 CYP3A4 (0.39) KDM4EKCNH2ALDH1A1POLBCHRM2
SCHEMBL9668463 0.80 ALDH1A1 (0.55) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9209326 0.80 KDM4E (0.42) KDM4EKCNH2ALDH1A1POLBCHRM2
SCHEMBL9147046 0.79 KDM4E (0.53) KDM4EKCNH2ALDH1A1POLBCHRM2
SCHEMBL9667565 0.79 KDM4E (0.72) KDM4EKCNH2ALDH1A1POLBTOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0388298-B1 Derivatives of pyridone carboxylic acids substituted by an azetidine, their preparation and their use as medicines ESTEVE LABOR DR (ES) 1995-06-21 EP claimed