SCHEMBL9212260

SCHEMBL9212260

CN1CCCC(CSc2nc3cccnc3s2)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.47
KCNH2 Q12809 4/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.37
CHRM1 P11229 4/20 0.36
CHRM2 P08172 3/20 0.36
ADRA2A P08913 2/20 0.36
DRD1 P21728 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
ADRA1A P35348 2/20 0.36
OPRM1 P35372 2/20 0.36
DRD3 P35462 2/20 0.36
HRH3 Q9Y5N1 2/20 0.36
CHRM3 P20309 2/20 0.36
HRH1 P35367 2/20 0.36
HTR6 P50406 2/20 0.36
ABCB11 O95342 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9215426 0.76 PDK1 (0.46) PDK1ADRA2A
SCHEMBL9215573 0.76 KCNH2 (0.38) PDK1KCNH2POLBCHRM1CHRM2
SCHEMBL9218698 0.73 PDK1 (0.54) PDK1ALDH1A1POLBHTR2CHTR1A
SCHEMBL9217289 0.73 PDK1 (0.50) PDK1ALDH1A1DRD1DRD3HRH3
SCHEMBL27550957 0.73 CRBN (0.43) KCNH2ALDH1A1POLBCHRM1CHRM2
SCHEMBL9275611 0.69 PDK1 (0.58) PDK1ALDH1A1POLBHTR2ACYP2D6
SCHEMBL9206848 0.68 PDK1 (0.50) PDK1ALDH1A1NPC1
SCHEMBL9208907 0.68 PDK1 (0.50) PDK1ALDH1A1POLBHTR2ALMNA
SCHEMBL9211341 0.67 PDK1 (0.59) PDK1ALDH1A1POLBLMNACYP2D6
SCHEMBL12090334 0.67 MAP4K4 (0.47) KCNH2CHRM1CHRM2ADRA2ADRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647231-A1 N-SUBSTITUTED 3-AZABICYCLO 3.2.0]HEPTANE DERIVATES USEFUL AS NEUROLEPTIC AGENTS, ETC. BASF AG (DE) 1995-04-12 EP disclosed
EP-0405976-B1 Azole derivatives and antiulcerative composition containing same MEIJI SEIKA CO (JP) 1995-04-05 EP disclosed
WO-1994000458-A1 N-SUBSTITUTED 3-AZABICYCLO[3.2.0]HEPTANE DERIVATES USEFUL AS NEUROLEPTIC AGENTS, ETC. BASF AKTIENGESELLSCHAFT (DE) 1994-01-06 WO disclosed
US-5200407-A Antisecretory agents MEIJI SEIKA KABURHIKI KAISHA (JP) 1993-04-06 US disclosed
US-5141946-A Antisecretory agents; acid resistance MEIJI SEIKA KABUSHIKI KAISHA (JP) 1992-08-25 US disclosed
US-5079255-A Nontoxic, acid stability MEIJI SEIKA KABUSHIKI KAISHA (JP) 1992-01-07 US disclosed