SCHEMBL9212875

SCHEMBL9212875

ClCCC1CCCCN1CCCc1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.47
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
SPHK2 Q9NRA0 2/20 0.39
SPHK1 Q9NYA1 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRNB1 P11230 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNB3 Q05901 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9208353 0.78 HRH3 (0.42) HRH3TDP1L3MBTL1CYP1A2CYP3A4
SCHEMBL27630471 0.78 OPRD1 (0.52) MEN1KMT2A
Hydrochloric Acid SCHEMBL9739345 0.77 HRH3 (0.40) HRH3TDP1L3MBTL1CYP1A2CYP3A4
SCHEMBL9216605 0.76 HRH3 (0.37) HRH3TDP1L3MBTL1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9739030 0.74 HRH3 (0.38) HRH3TDP1L3MBTL1CYP1A2CYP3A4
SCHEMBL9215931 0.73 HRH3 (0.38) HRH3TDP1L3MBTL1CYP1A2CYP3A4
SCHEMBL5888846 0.73
SCHEMBL8542041 0.73 CYP19A1 (0.45) CYP1A2CYP3A4
SCHEMBL9820990 0.73 SIGMAR1 (0.47)
SCHEMBL9205342 0.73 KDM4E (0.38) HRH3TDP1L3MBTL1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed