SCHEMBL9212951

SCHEMBL9212951

COc1cc2c(cc1OC)C(=O)N(CC1CCCN(CCc3ccc([N+](=O)[O-])cc3)C1)C2

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.47
ABCG2 Q9UNQ0 3/20 0.47
ACHE P22303 2/20 0.47
BCHE P06276 1/20 0.47
KCNJ1 P48048 3/20 0.45
KCNH2 Q12809 3/20 0.45
HRH3 Q9Y5N1 3/20 0.44
ABCC1 P33527 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9213616 0.99 ABCB1 (0.47) ABCB1ABCG2ACHEBCHEKCNJ1
SCHEMBL9216056 0.89 BCHE (0.44) ACHEBCHE
SCHEMBL9212603 0.89 GAA (0.50) ABCB1HRH3
SCHEMBL9212017 0.88 GAA (0.46)
SCHEMBL9208083 0.88 ABCB1 (0.44) ABCB1ABCG2
Hydrochloric Acid SCHEMBL9212998 0.87 ABCB1 (0.44) ABCB1ABCG2
SCHEMBL9739245 0.86 ABCG2 (0.51) ABCB1ABCG2ACHEBCHEKCNJ1
SCHEMBL9207120 0.85 ACHE (0.47) ACHEBCHE
SCHEMBL9213519 0.85 GAA (0.40) ACHE
Hydrochloric Acid SCHEMBL9740859 0.85 ABCG2 (0.50) ABCB1ABCG2ACHEBCHEKCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed