SCHEMBL9208083

SCHEMBL9208083

COc1cc2c(cc1OC)C(=O)N(CC1CCCN(CCc3ccc(N)cc3)C1)C2

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.44
ABCG2 Q9UNQ0 2/20 0.44
GAA P10253 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CNR2 P34972 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9212998 0.99 ABCB1 (0.44) ABCB1ABCG2GAAMEN1KMT2A
SCHEMBL9216056 0.92 BCHE (0.44) GAAMEN1KMT2ACHRNB2CHRNB4
SCHEMBL9212603 0.92 GAA (0.50) ABCB1GAAMEN1KMT2A
SCHEMBL9212017 0.91 GAA (0.46) GAAMEN1KMT2ACNR2CHRNB2
SCHEMBL9207120 0.89 ACHE (0.47) GAAMEN1KMT2ACHRNB2CHRNB4
SCHEMBL9213519 0.88 GAA (0.40) GAAMEN1KMT2ACHRNB2CHRNB4
SCHEMBL9212951 0.88 ABCB1 (0.47) ABCB1ABCG2
SCHEMBL9215835 0.88 SIGMAR1 (0.46) GAAMEN1KMT2A
Hydrochloric Acid SCHEMBL9207786 0.87 DHCR7 (0.43) GAAMEN1KMT2A
SCHEMBL9213493 0.87 MEN1 (0.41) GAAMEN1KMT2ACHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed