SCHEMBL9212975

SCHEMBL9212975

Cc1cc2c(cc1C)CC(=O)N(CC1CCCN(CCCCCc3cccs3)C1)CC2

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.35
HTR7 P34969 3/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 2/20 0.33
LTA4H P09960 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HTR1A P08908 1/20 0.33
KCNH2 Q12809 1/20 0.32
GHSR Q92847 1/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9208876 0.99 HRH3 (0.36) HRH3HTR7ALDH1A1KDM4ELMNA
SCHEMBL9207422 0.93 HRH3 (0.40) HRH3ALDH1A1KDM4ELMNALTA4H
SCHEMBL9208037 0.91 HRH3 (0.37) HRH3ALDH1A1KDM4ELMNALTA4H
Hydrochloric Acid SCHEMBL9740263 0.90 ALOX15 (0.42) ALDH1A1KDM4EHTR1AKCNH2GAA
Hydrochloric Acid SCHEMBL9739549 0.90 ALOX15 (0.42) ALDH1A1KDM4EHTR1AKCNH2GAA
SCHEMBL9206630 0.90 ALOX15 (0.43) ALDH1A1KDM4EHTR1AKCNH2GAA
SCHEMBL9208761 0.90 NPC1 (0.35) HRH3HTR7ALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL9740340 0.89 ALOX15 (0.43) ALDH1A1KDM4EHTR1AKCNH2GAA
SCHEMBL9206564 0.89 NPC1 (0.36) HRH3HTR7ALDH1A1KDM4ELMNA
SCHEMBL9216033 0.88 ATM (0.39) HRH3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed