SCHEMBL9213580

SCHEMBL9213580

NCC(=O)C(O[C]=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
GABBR2 O75899 1/20 0.40
GABBR1 Q9UBS5 1/20 0.40
SLC6A3 Q01959 3/20 0.38
LMNA P02545 3/20 0.38
DRD3 P35462 2/20 0.38
MAPK1 P28482 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
EDNRB P24530 1/20 0.38
MC4R P32245 1/20 0.38
CYP2C19 P33261 1/20 0.38
MC3R P41968 1/20 0.38
DRD2 P14416 1/20 0.38
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11211550 0.83 ALDH1A1 (0.40) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL11095898 0.81 CNR2 (0.44) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL710572 0.80 CYP2D6 (0.46) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
Ethylene SCHEMBL29161565 0.79 GABBR2 (0.42) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL9068581 0.77 ALDH1A1 (0.51) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL5157376 0.75 ALDH1A1 (0.64) CYP1A2SMN1; SMN2NPSR1ALDH1A1CYP3A4
SCHEMBL1371273 0.75 MMP8 (0.50) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL712324 0.74 KMT2A (0.56) PKMSMN1; SMN2ALDH1A1CYP3A4LMNA
SCHEMBL212215 0.73 ALDH1A1 (0.51) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL19551413 0.73 KLK7 (0.54) SMN1; SMN2ALDH1A1GAAEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295316-B1 Antitumor amino acid and peptide derivatives of 1,4-bis[ (aminoalkyl and hydroxyaminoalkyl)- amino]-5,8 dihydroxyanthraquinones AMERICAN CYANAMID CO (US) 1995-11-08 EP disclosed
EP-0489220-A1 Cytotoxic N,N'-bis (succinyl-peptide-) derivatives of 1,4-bis (aminoalkyl)-5,8-dihydroxyanthraquinones and antibody conjugates thereof AMERICAN CYANAMID COMPANY (US) 1992-06-10 EP disclosed