SCHEMBL9217834

SCHEMBL9217834

CCCn1nnc(-c2cnc3cccc(C)n3c2=O)n1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.36
RAB9A P51151 6/20 0.35
SMN1; SMN2 Q16637 6/20 0.35
NPC1 O15118 4/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
ATM Q13315 1/20 0.34
ALOX15 P16050 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
USP2 O75604 1/20 0.33
CYP2C9 P11712 1/20 0.33
TOP2A P11388 1/20 0.32
QPCT Q16769 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9259873 0.92 TRPV1 (0.38)
SCHEMBL9208224 0.91 SMN1; SMN2 (0.39) HTTSMN1; SMN2TSHRALDH1A1LMNA
SCHEMBL9217990 0.80 NPC1 (0.39) HTTRAB9ASMN1; SMN2NPC1TSHR
SCHEMBL9213645 0.79 HTT (0.37) HTTRAB9ANPC1ALDH1A1CYP1A2
SCHEMBL9255169 0.78 CYP1A2 (0.43) HTTSMN1; SMN2ALDH1A1CYP1A2CYP2C19
SCHEMBL9210936 0.74 MAPT (0.40) HTTRAB9ASMN1; SMN2NPC1TSHR
SCHEMBL9210655 0.74 TP53 (0.39) ALDH1A1NPSR1MAPTLMNAHPGD
Hydrochloric Acid SCHEMBL9219227 0.73 TP53 (0.39) ALDH1A1NPSR1MAPTLMNAHPGD
SCHEMBL9259026 0.73 ADORA2A (0.38) HTTALDH1A1CYP1A2CYP2C19MAPT
SCHEMBL9263794 0.73 HTT (0.40) HTTSMN1; SMN2ALDH1A1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475000-A Antiulcer agents CHINOIN GYOGYSZER-ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1995-12-12 US disclosed
EP-0641340-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO- 1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1995-03-08 EP disclosed
WO-1993004065-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO-[1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-03-04 WO disclosed