SCHEMBL9213867

SCHEMBL9213867

CNC(=O)Nc1ccc(/C=C/CC(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAM P19021 1/20 0.54
MAOB P27338 4/20 0.50
ALDH1A1 P00352 5/20 0.49
KMT2A Q03164 4/20 0.44
NPC1 O15118 5/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MAOA P21397 3/20 0.42
POLB P06746 1/20 0.41
MEN1 O00255 3/20 0.40
CYP3A4 P08684 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MAPT P10636 3/20 0.40
CYP4F2 P78329 1/20 0.39
CYP4A11 Q02928 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210792 0.85 PAM (0.51) PAMMAOBALDH1A1KMT2ARAB9A
SCHEMBL8868330 0.84 ALDH1A1 (0.51) MAOBALDH1A1KMT2ANPC1RAB9A
SCHEMBL8868345 0.84 ALDH1A1 (0.51) MAOBALDH1A1KMT2ANPC1RAB9A
SCHEMBL8868335 0.84 ALDH1A1 (0.51) MAOBALDH1A1KMT2ANPC1RAB9A
SCHEMBL8828409 0.84 PAM (0.58) PAMMAOBALDH1A1KMT2ANPC1
SCHEMBL8828415 0.84 PAM (0.58) PAMMAOBALDH1A1KMT2ANPC1
SCHEMBL7746675 0.79 ALDH1A1 (0.53) MAOBALDH1A1KMT2ANPC1RAB9A
SCHEMBL7746671 0.79 ALDH1A1 (0.53) MAOBALDH1A1KMT2ANPC1RAB9A
SCHEMBL9155176 0.78 MAPT (0.45) PAMMAOBALDH1A1KMT2ANPC1
SCHEMBL9155171 0.78 MAPT (0.45) PAMMAOBALDH1A1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0399358-B1 Butenoic acid derivatives EISAI CO LTD (JP) 1995-03-08 EP disclosed
EP-0633248-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1995-01-11 EP disclosed
EP-0589491-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1994-03-30 EP disclosed