SCHEMBL9215200

SCHEMBL9215200

CC=C(C(=O)O)c1csc2ccc(CN(C)C(C)c3ccccc3)cc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GCGR P47871 1/20 0.38
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TBXAS1 P24557 1/20 0.35
FFAR2 O15552 2/20 0.35
MAPK14 Q16539 1/20 0.35
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
TSHR P16473 1/20 0.34
C5AR1 P21730 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
ADAM17 P78536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213989 0.91 GCGR (0.37) GCGRMEN1KMT2AKDM4ETBXAS1
SCHEMBL9215196 0.91 GCGR (0.35) GCGRMEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL9213982 0.85 GCGR (0.36) GCGRMEN1KMT2AKDM4ETBXAS1
SCHEMBL9312641 0.67 TBXAS1 (0.37) MEN1KMT2AKDM4ESMN1; SMN2TBXAS1
SCHEMBL9313258 0.67 FFAR1 (0.48) MEN1KMT2ASMN1; SMN2
SCHEMBL8027272 0.66 HTR2A (0.60) KDM4EOPRK1TSHRALDH1A1
SCHEMBL18055963 0.66 HTR2A (0.60) KDM4EOPRK1TSHRALDH1A1
SCHEMBL6837412 0.66 HTR2A (0.60) KDM4EOPRK1TSHRALDH1A1
SCHEMBL9218481 0.62 PTK2 (0.38) MEN1KMT2AKDM4ETBXAS1
SCHEMBL9218877 0.61 HDAC3 (0.54) MEN1KMT2AKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433233-B1 Heterocyclic compounds CIBA GEIGY AG (CH) 1995-01-25 EP claimed