SCHEMBL9215501

SCHEMBL9215501

CCc1ncnc(NC(CC)c2ccc(OC(F)(F)Br)cc2)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.36
RPS6KB1 P23443 2/20 0.36
AURKA O14965 1/20 0.36
PDPK1 O15530 1/20 0.36
AKT1 P31749 3/20 0.35
CRHR1 P34998 2/20 0.34
PDE2A O00408 5/20 0.32
PDE3A Q14432 1/20 0.32
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216328 0.92 AURKA (0.42) EGFRRPS6KB1AURKAPDPK1AKT1
SCHEMBL9523428 0.90 EGFR (0.36) EGFRRPS6KB1AURKAPDPK1AKT1
SCHEMBL9524057 0.86 EGFR (0.36) EGFRRPS6KB1AURKAPDPK1AKT1
SCHEMBL9193841 0.84 CRHR1 (0.39) EGFRRPS6KB1AKT1CRHR1
SCHEMBL9084666 0.83 PTGER4 (0.40) EGFRRPS6KB1AURKACRHR1
Hydrochloric Acid SCHEMBL9523871 0.82 PTGER4 (0.39) EGFRRPS6KB1AURKACRHR1
SCHEMBL9523756 0.82 CRHR1 (0.39) EGFRRPS6KB1AURKAAKT1CRHR1
SCHEMBL9212072 0.81 EGFR (0.36) EGFRRPS6KB1AKT1CRHR1
SCHEMBL8303141 0.81 EGFR (0.38) EGFRRPS6KB1AKT1CRHR1
SCHEMBL9212840 0.81 ALDH1A1 (0.35) EGFRRPS6KB1AURKAPDPK1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5141941-A ARALKYLAMINE DERIVATIVES, AND FUNGICIDES CONTAINING THE SAME UBE INDUSTRIES, LTD. (JP) 1992-08-25 US claimed
EP-0370704-B1 Aralkylamine derivatives, preparation thereof and fungicides containing the same UBE INDUSTRIES (JP) 1995-02-01 EP disclosed
US-5141941-A ARALKYLAMINE DERIVATIVES, AND FUNGICIDES CONTAINING THE SAME UBE INDUSTRIES, LTD. (JP) 1992-08-25 US disclosed
EP-0370704-A2 Aralkylamine derivatives, preparation thereof and fungicides containing the same UBE INDUSTRIES, LTD. (JP) 1990-05-30 EP disclosed