SCHEMBL9215967

SCHEMBL9215967

O=C1Cc2cc3c(cc2CCN1CC1CCN(CCc2cc4ccccc4o2)C1)OCO3

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 6/20 0.38
DRD2 P14416 3/20 0.36
ACHE P22303 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
MAPK1 P28482 1/20 0.34
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217026 0.95 MAPK1 (0.40) HTR2BDRD2ALDH1A1MAPK1
SCHEMBL9207626 0.94 MAPK1 (0.38) HTR2BDRD2ALDH1A1MAPK1
SCHEMBL9207136 0.90 HTR2B (0.39) HTR2BDRD2ACHESLC6A4SLC6A3
SCHEMBL9208812 0.90 DRD2 (0.38) HTR2BDRD2ALDH1A1MAPK1
SCHEMBL9209357 0.89 DRD2 (0.37) HTR2BDRD2ALDH1A1MAPK1
SCHEMBL9216985 0.87 HTR2B (0.45) HTR2BDRD2ACHEALDH1A1SLC6A4
SCHEMBL9215152 0.85 MAPK1 (0.44) HTR2BDRD2MAPK1
SCHEMBL9213117 0.84 MAPK1 (0.42) HTR2BDRD2MAPK1
SCHEMBL9207394 0.83 HCRTR1 (0.44) HTR2BDRD2ACHEMAPK1HTR1A
SCHEMBL9210489 0.82 HCRTR1 (0.44) HTR2BDRD2ACHEALDH1A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed